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Discovery of Novel and Long Acting Muscarinic Acetylcholine Receptor AntagonistsJIAN JIN; YONGHUI WANG; BERLANGA, Manuela et al.Journal of medicinal chemistry (Print). 2008, Vol 51, Num 16, pp 4866-4869, issn 0022-2623, 4 p.Article

2' Biaryl amides as novel and subtype selective M1 agonists. Part II: Further optimization and profilingBUDZILC, Brian; GARZYA, Vincenzo; FORBES, Ian T et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 12, pp 3545-3549, issn 0960-894X, 5 p.Article

Potent and selective small-molecule human urotensin-II antagonists with improved pharmacokinetic profilesMCATEE, John J; DODSON, Jason W; DONGCHUAN SHI et al.Bioorganic & medicinal chemistry letters (Print). 2008, Vol 18, Num 13, pp 3716-3719, issn 0960-894X, 4 p.Article

Muscarinic acetylcholine receptor antagonists : SAR and optimization of tyrosine ureasJIAN JIN; YONGHUI WANG; MOORE, Michael L et al.Bioorganic & medicinal chemistry letters (Print). 2008, Vol 18, Num 20, pp 5481-5486, issn 0960-894X, 6 p.Article

Phenoxyacetic acids as PPARδ partial agonists: Synthesis, optimization, and in vivo efficacyEVANS, Karen A; SHEARER, Barry G; EPPERLY, Andrea H et al.Bioorganic & medicinal chemistry letters (Print). 2011, Vol 21, Num 8, pp 2345-2350, issn 0960-894X, 6 p.Article

2-Aminomethyl piperidines as novel urotensin-II receptor antagonistsJIAN JIN; YONGHUI WANG; VAIDYA, Kalindi S et al.Bioorganic & medicinal chemistry letters (Print). 2008, Vol 18, Num 9, pp 2860-2864, issn 0960-894X, 5 p.Article

2' Biaryl amides as novel and subtype selective M1 agonists. Part I: Identification, synthesis, and initial SARBUDZIK, Brian; GARZYA, Vincenzo; DONGCHUAN SHI et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 12, pp 3540-3544, issn 0960-894X, 5 p.Article

Structure―activity relationship studies of novel 3-oxazolidinedione-6-naphthyl-2-pyridinones as potent and orally bioavailable EP3 receptor antagonistsMORALES-RAMOS, Angel I; LI, Yue H; JAWORSKI, Jon-Paul et al.Bioorganic & medicinal chemistry letters (Print). 2011, Vol 21, Num 10, pp 2806-2811, issn 0960-894X, 6 p.Article

M3 muscarinic acetylcholine receptor antagonists : SAR and optimization of bi-aryl aminesBUDZIK, Brian; YONGHUI WANG; SARAU, Henry M et al.Bioorganic & medicinal chemistry letters (Print). 2009, Vol 19, Num 6, pp 1686-1690, issn 0960-894X, 5 p.Article

Discovery of Biphenyl Piperazines as Novel and Long Acting Muscarinic Acetylcholine Receptor AntagonistsJIAN JIN; BUDZIK, Brian; BERLANGA, Manuela et al.Journal of medicinal chemistry (Print). 2008, Vol 51, Num 19, pp 5915-5918, issn 0022-2623, 4 p.Article

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